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  • 1-10 ل  90,730 نتائج ل ""proteolysis""
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Academic Journal

Discovery of a Proteolysis Targeting Chimera for TRKA and RET-derived oncoproteins.

  • Authors : Moccia M; Istituto degli Endotipi in Oncologia, Metabolismo e Immunologia 'G. Salvatore' (IEOMI) del CNR, Naples, Italia.; Zhang L

Subjects: Proto-Oncogene Proteins c-ret*/Proto-Oncogene Proteins c-ret*/Proto-Oncogene Proteins c-ret*/metabolism ; Proto-Oncogene Proteins c-ret*/Proto-Oncogene Proteins c-ret*/Proto-Oncogene Proteins c-ret*/antagonists & inhibitors ; Proto-Oncogene Proteins c-ret*/Proto-Oncogene Proteins c-ret*/Proto-Oncogene Proteins c-ret*/genetics

  • Source: Scientific reports [Sci Rep] 2025 Nov 25; Vol. 15 (1), pp. 41770. Date of Electronic Publication: 2025 Nov 25.Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101563288 Publication Model: Electronic Cited Medium: Internet ISSN:

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Academic Journal

Design and Synthesis of Novel Candidate CK1δ Proteolysis Targeting Chimeras (PROTACs).

  • Authors : Arnold M; Institute of Pharmacy, Department of Pharmaceutical and Medicinal Chemistry, Christian-Albrechts-University of Kiel, 24118 Kiel, Germany.; Thompson T

Subjects: Proteolysis*/Proteolysis*/Proteolysis*/drug effects ; Casein Kinase Idelta*/Casein Kinase Idelta*/Casein Kinase Idelta*/antagonists & inhibitors ; Casein Kinase Idelta*/Casein Kinase Idelta*/Casein Kinase Idelta*/metabolism

  • Source: Molecules (Basel, Switzerland) [Molecules] 2025 Nov 18; Vol. 30 (22). Date of Electronic Publication: 2025 Nov 18.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Targeting Protein Tyrosine Phosphatases via PROteolysis-TArgeting Chimeras (PROTACs): Current Developments and Prospects.

  • Authors : Maccari R; Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina, Viale F. Stagno d'Alcontres 31, 98166 Messina, Italy.

Subjects: Proteolysis*/Proteolysis*/Proteolysis*/drug effects ; Protein Tyrosine Phosphatases*/Protein Tyrosine Phosphatases*/Protein Tyrosine Phosphatases*/antagonists & inhibitors ; Protein Tyrosine Phosphatases*/Protein Tyrosine Phosphatases*/Protein Tyrosine Phosphatases*/metabolism

  • Source: Molecules (Basel, Switzerland) [Molecules] 2025 Nov 18; Vol. 30 (22). Date of Electronic Publication: 2025 Nov 18.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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  • 1-10 ل  90,730 نتائج ل ""proteolysis""