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Academic Journal

Design and Evaluation of Indole-Based Schiff Bases as α-Glucosidase Inhibitors: CNN-Enhanced Docking, MD Simulations, ADMET Profiling, and SAR Analysis.

  • Authors : Bhagwat SK; Department of Chemistry, Research Centre HPT Arts, RYK Science College (Affiliated to S. P. Pune University), Nashik 422005, Maharashtra, India.; Patil SV

Subjects: Glycoside Hydrolase Inhibitors*/Glycoside Hydrolase Inhibitors*/Glycoside Hydrolase Inhibitors*/chemistry ; Glycoside Hydrolase Inhibitors*/Glycoside Hydrolase Inhibitors*/Glycoside Hydrolase Inhibitors*/pharmacology ; Glycoside Hydrolase Inhibitors*/Glycoside Hydrolase Inhibitors*/Glycoside Hydrolase Inhibitors*/chemical synthesis

  • Source: Molecules (Basel, Switzerland) [Molecules] 2025 Sep 08; Vol. 30 (17). Date of Electronic Publication: 2025 Sep 08.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Polymorph Selection and Derivatization in Enantiomerically Pure Medicarpin: Crystallographic and Computational Insights.

  • Authors : Guevara-Martínez SJ; Department of Pharmacology, School of Exact Sciences and Engineering, University of Guadalajara, Boulevard Gral. Marcelino García Barragán 1421, Olímpica, Guadalajara 44430, Jalisco, Mexico.; Herrera-Bucio R

  • Source: Molecules (Basel, Switzerland) [Molecules] 2025 Sep 08; Vol. 30 (17). Date of Electronic Publication: 2025 Sep 08.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Morphology-Dependent Transformation of Dicalcium Phosphate Dihydrate (DCPD) to Octacalcium Phosphate (OCP) and Its Stability in Simulated Physiological Fluids.

  • Authors : Chávez-Herrera D; Unidad Profesional Interdisciplinaria de Ingeniería Campus Guanajuato, Instituto Politécnico Nacional, Guanajuato 36275, Mexico.; Rangel-Villanueva E

Subjects: Calcium Phosphates*/Calcium Phosphates*/Calcium Phosphates*/chemistry ; Body Fluids*/Body Fluids*/Body Fluids*/chemistry; X-Ray Diffraction

  • Source: Molecules (Basel, Switzerland) [Molecules] 2025 Sep 05; Vol. 30 (17). Date of Electronic Publication: 2025 Sep 05.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Synergistic Disruption of Foodborne Pathogen Biofilms by Oregano Essential Oil and Bacteriophage phiLLS: Atomic Force Microscopy Insights.

Subjects: Biofilms*/Biofilms*/Biofilms*/drug effects ; Biofilms*/Biofilms*/Biofilms*/growth & development ; Oils, Volatile*/Oils, Volatile*/Oils, Volatile*/pharmacology

  • Source: Molecules (Basel, Switzerland) [Molecules] 2025 Aug 30; Vol. 30 (17). Date of Electronic Publication: 2025 Aug 30.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Photoprotective Effect of Annona muricata L. Extracts in Rats Exposed to Ultraviolet Radiation via P53 and RB Gene Expression.

Subjects: Plant Extracts*/Plant Extracts*/Plant Extracts*/pharmacology ; Plant Extracts*/Plant Extracts*/Plant Extracts*/chemistry ; Annona*/Annona*/Annona*/chemistry

  • Source: Molecules (Basel, Switzerland) [Molecules] 2025 Aug 28; Vol. 30 (17). Date of Electronic Publication: 2025 Aug 28.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

A Comprehensive Review of Niosomes: Composition, Structure, Formation, Characterization, and Applications in Bioactive Molecule Delivery Systems.

  • Authors : Bautista-Solano AA; Departamento de Ingeniería Bioquímica, Escuela Nacional de Ciencias Biológicas, Instituto Politécnico Nacional (IPN), Av. Wilfrido Massieu Esq. Miguel Stampa s/n, Zacatenco, Alcaldía Gustavo A. Madero, Ciudad de Mexico 07728, Mexico.; Dávila-Ortiz G

Subjects: Liposomes*/Liposomes*/Liposomes*/chemistry ; Drug Delivery Systems* ; Drug Carriers*/Drug Carriers*/Drug Carriers*/chemistry

  • Source: Molecules (Basel, Switzerland) [Molecules] 2025 Aug 23; Vol. 30 (17). Date of Electronic Publication: 2025 Aug 23.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Semi-Synthesis, Anti-Leukemia Activity, and Docking Study of Derivatives from 3 α ,24-Dihydroxylup-20(29)-en-28-Oic Acid.

  • Authors : Noh-Burgos MJ; Unidad de Biotecnología, Centro de Investigación Científica de Yucatán (CICY), Mérida 97205, Mexico.; Unidad Médica de Alta Especialidad, Centro Médico Ignacio García Téllez, Instituto Mexicano del Seguro Social (IMSS), Mérida 97200, Mexico.

Subjects: Molecular Docking Simulation* ; Antineoplastic Agents*/Antineoplastic Agents*/Antineoplastic Agents*/pharmacology ; Antineoplastic Agents*/Antineoplastic Agents*/Antineoplastic Agents*/chemical synthesis

  • Source: Molecules (Basel, Switzerland) [Molecules] 2025 Jul 30; Vol. 30 (15). Date of Electronic Publication: 2025 Jul 30.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Quercetin Reduces Antinociceptive but Not the Anti-Inflammatory Effects of Indomethacin, Ketorolac, and Celecoxib in Rats with Gout-like Pain.

  • Authors : Aviles-Herrera J; Departamento de Farmacología, Facultad de Medicina, Universidad Nacional Autónoma de México (UNAM), Ciudad de México 04510, Mexico.; Ángeles-López GE

  • Source: Molecules (Basel, Switzerland) [Molecules] 2025 Jul 30; Vol. 30 (15). Date of Electronic Publication: 2025 Jul 30.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Immunometabolic Effects of Ginger ( Zingiber officinale Roscoe) Supplementation in Obesity: A Comprehensive Review.

  • Authors : Preciado-Ortiz ME; Institute of Translational Nutrigenetics and Nutrigenomics, Department of Molecular Biology and Genomics, University Center of Health Sciences, University of Guadalajara, Guadalajara 44340, Jalisco, Mexico.; Gembe-Olivarez G

Subjects: Zingiber officinale*/Zingiber officinale*/Zingiber officinale*/chemistry ; Obesity*/Obesity*/Obesity*/drug therapy ; Obesity*/Obesity*/Obesity*/metabolism

  • Source: Molecules (Basel, Switzerland) [Molecules] 2025 Jul 11; Vol. 30 (14). Date of Electronic Publication: 2025 Jul 11.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Antimicrobial Activity of Cinnamon, Tea Tree, and Thyme Essential Oils Against Pathogenic Bacteria Isolated from Tilapia ( Oreochromis spp.) in Aquaculture Farms.

  • Authors : Terrazas-Pineda KA; Departamento de Ingeniería Bioquímica, Escuela Nacional de Ciencias Biológicas, Instituto Politécnico Nacional, Unidad Profesional Adolfo López Mateos, Zacatenco, Av. Wilfrido Massieu 399, Col. Nueva Industrial Vallejo, Alcaldía Gustavo A. Madero, Ciudad de México CP 07738, Mexico.; Alamilla-Beltrán L

Subjects: Thymus Plant*/Thymus Plant*/Thymus Plant*/chemistry ; Oils, Volatile*/Oils, Volatile*/Oils, Volatile*/pharmacology ; Oils, Volatile*/Oils, Volatile*/Oils, Volatile*/chemistry

  • Source: Molecules (Basel, Switzerland) [Molecules] 2025 Jun 28; Vol. 30 (13). Date of Electronic Publication: 2025 Jun 28.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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