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  • 1-10 ل  5,377 نتائج ل ""Binding, Competitive""
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Academic Journal

Vibrio splendidus infection promotes circRNA-FGL1-regulated coelomocyte apoptosis via competitive binding to Myc with the deubiquitinase OTUB1 in Apostichopus japonicus.

  • Authors : Guo M; State Key Laboratory for Managing Biotic and Chemical Threats to the Quality and Safety of Agro-products, School of Marine Sciences, Ningbo University, Ningbo, China.; Li X

Subjects: Apoptosis* ; RNA, Circular*/RNA, Circular*/RNA, Circular*/metabolism ; RNA, Circular*/RNA, Circular*/RNA, Circular*/genetics Vibrio splendidus

  • Source: PLoS pathogens [PLoS Pathog] 2024 Aug 15; Vol. 20 (8), pp. e1012463. Date of Electronic Publication: 2024 Aug 15 (Print Publication: 2024).Publisher: Public Library of Science Country of Publication: United States NLM ID: 101238921 Publication Model: eCollection Cited Medium: Internet

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Academic Journal

A novel and selective fluorescent ligand for the study of adenosine A 2B receptors.

  • Authors : Patera F; Division of Physiology, Pharmacology and Neuroscience, School of Life Sciences, University of Nottingham, Nottingham, UK.; Centre of Membrane Proteins and Receptors (COMPARE), University of Birmingham and University of Nottingham, Midlands, UK.

Subjects: Receptor, Adenosine A2B*/Receptor, Adenosine A2B*/Receptor, Adenosine A2B*/metabolism ; Fluorescent Dyes*/Fluorescent Dyes*/Fluorescent Dyes*/chemistry ; Macrophages*/Macrophages*/Macrophages*/metabolism

  • Source: Pharmacology research & perspectives [Pharmacol Res Perspect] 2024 Aug; Vol. 12 (4), pp. e1223.Publisher: John Wiley & Sons Ltd, British Pharmacological Society and American Society for Pharmacology and Experimental Therapeutics Country of Publication: United States

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Academic Journal

Theory on the rate equations of Michaelis-Menten type enzyme kinetics with competitive inhibition.

  • Authors : Murugan R; Department of Biotechnology, Indian Institute of Technology Madras, Chennai, Tamil Nadu, India.

Subjects: Enzymes*/Enzymes*/Enzymes*/metabolism ; Enzyme Inhibitors*/Enzyme Inhibitors*/Enzyme Inhibitors*/pharmacology; Kinetics

  • Source: PloS one [PLoS One] 2024 Jul 18; Vol. 19 (7), pp. e0302679. Date of Electronic Publication: 2024 Jul 18 (Print Publication: 2024).Publisher: Public Library of Science Country of Publication: United States NLM ID: 101285081 Publication Model: eCollection Cited Medium: Internet

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Academic Journal

Discovery of Novel Delta Opioid Receptor (DOR) Inverse Agonist and Irreversible (Non-Competitive) Antagonists.

  • Authors : Tanguturi P; Department of Pharmacology, College of Medicine, University of Arizona, Tucson, AZ 85724, USA.; Pathak V

Subjects: Binding, Competitive* ; Drug Discovery*/Drug Discovery*/Drug Discovery*/methods; Analgesics, Opioid/Analgesics, Opioid/Analgesics, Opioid/*chemistry

  • Source: Molecules (Basel, Switzerland) [Molecules] 2021 Nov 05; Vol. 26 (21). Date of Electronic Publication: 2021 Nov 05.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Removal of Protein-Bound Uremic Toxins Using Binding Competitors in Hemodialysis: A Narrative Review.

Subjects: Binding, Competitive* ; Renal Dialysis*; Dialysis Solutions/Dialysis Solutions/Dialysis Solutions/*chemistry

  • Source: Toxins [Toxins (Basel)] 2021 Sep 04; Vol. 13 (9). Date of Electronic Publication: 2021 Sep 04.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101530765 Publication Model: Electronic Cited Medium: Internet ISSN: 2072-6651

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Academic Journal

An Integrated Approach toward NanoBRET Tracers for Analysis of GPCR Ligand Engagement.

  • Authors : Killoran MP; Promega Corporation, 2800 Woods Hollow, Fitchburg, WI 53711, USA.; Levin S

Subjects: Binding, Competitive* ; Machine Learning*; Bioluminescence Resonance Energy Transfer Techniques/Bioluminescence Resonance Energy Transfer Techniques/Bioluminescence Resonance Energy Transfer Techniques/*methods

  • Source: Molecules (Basel, Switzerland) [Molecules] 2021 May 12; Vol. 26 (10). Date of Electronic Publication: 2021 May 12.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Synthesis of a Coumarin-Based PPARγ Fluorescence Probe for Competitive Binding Assay.

  • Authors : Yoshikawa C; Laboratory of Drug Design and Medicinal Chemistry, Showa Pharmaceutical University, 3-3165 Higashi-Tamagawagakuen, Machida, Tokyo 194-8543, Japan.; Ishida H

Subjects: Binding, Competitive* ; Biological Assay*; Coumarins/Coumarins/Coumarins/*chemistry

  • Source: International journal of molecular sciences [Int J Mol Sci] 2021 Apr 14; Vol. 22 (8). Date of Electronic Publication: 2021 Apr 14.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

Inhibitors in AKTion: ATP-competitive vs allosteric.

  • Authors : Lazaro G; Division of Cancer Therapeutics, The Institute of Cancer Research, 15 Cotswold Rd., SM2 5NG London, U.K.; Kostaras E

Subjects: Allosteric Site* ; Binding, Competitive* ; Gene Expression Regulation, Neoplastic*

  • Source: Biochemical Society transactions [Biochem Soc Trans] 2020 Jun 30; Vol. 48 (3), pp. 933-943.Publisher: Portland Press On The Behalf Of The Biochemical Society Country of Publication: England NLM ID: 7506897 Publication Model: Print Cited Medium:

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Academic Journal

Higher naloxone dosing in a quantitative systems pharmacology model that predicts naloxone-fentanyl competition at the opioid mu receptor level.

  • Authors : Moss RB; Adamis Pharmaceuticals Corp, San Diego, CA, United States of America.; Pryor MM

Subjects: Binding, Competitive* ; Models, Theoretical*; Fentanyl/Fentanyl/Fentanyl/*metabolism

  • Source: PloS one [PLoS One] 2020 Jun 16; Vol. 15 (6), pp. e0234683. Date of Electronic Publication: 2020 Jun 16 (Print Publication: 2020).Publisher: Public Library of Science Country of Publication: United States NLM ID: 101285081 Publication Model: eCollection Cited Medium: Internet

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Academic Journal

Identifying neural substrates of competitive interactions and sequence transitions during mechanosensory responses in Drosophila.

  • Authors : Masson JB; Janelia Research Campus, Howard Hughes Medical Institute, Ashburn, Virginia, United States of America.; Decision and Bayesian Computation, USR 3756 (C3BI/DBC) & Neuroscience Department, Institut Pasteur & CNRS, Paris, France.

Subjects: Binding, Competitive*/Binding, Competitive*/Binding, Competitive*/physiology; Action Potentials/Action Potentials/Action Potentials/*physiology ; Mechanotransduction, Cellular/Mechanotransduction, Cellular/Mechanotransduction, Cellular/*physiology

  • Source: PLoS genetics [PLoS Genet] 2020 Feb 14; Vol. 16 (2), pp. e1008589. Date of Electronic Publication: 2020 Feb 14 (Print Publication: 2020).Publisher: Public Library of Science Country of Publication: United States NLM ID: 101239074 Publication Model: eCollection Cited Medium: Internet

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  • 1-10 ل  5,377 نتائج ل ""Binding, Competitive""