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Academic Journal

Virtual Screening of Novel Benzothiozinone Derivatives to Predict Potential Inhibitors of Mycobacterium Tuberculosis Kinases 2D-QSAR, Molecular Docking, MM-PBSA Dynamics Simulations, and ADMET Properties.

  • Authors : Guendouzi A; Higher Normal School of Constantine ENS Assia Djebar Constantine, Ali Mendjeli, Constantine 25000, Algeria.; Pharmaceutical Sciences Research Center CRSP, ZAM Ali Mendjeli, Constantine 25000, Algeria.

Subjects: Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/enzymology ; Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/drug effects ; Antitubercular Agents*/Antitubercular Agents*/Antitubercular Agents*/chemistry

  • Source: International journal of molecular sciences [Int J Mol Sci] 2025 May 27; Vol. 26 (11). Date of Electronic Publication: 2025 May 27.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

Efficacy and immunogenicity of rKVAC85B in a BCG prime-boost regimen against H37Rv and HN878 Mycobacterium tuberculosis strains.

  • Authors : Shin E; National Institute of Infectious Diseases, National Institute of Health, Korea Disease Control and Prevention Agency, CheongJu, Chungbuk, Republic of Korea.; Yun JS

Subjects: Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/immunology ; Antigens, Bacterial*/Antigens, Bacterial*/Antigens, Bacterial*/immunology ; Antigens, Bacterial*/Antigens, Bacterial*/Antigens, Bacterial*/genetics

  • Source: PloS one [PLoS One] 2025 May 14; Vol. 20 (5), pp. e0322147. Date of Electronic Publication: 2025 May 14 (Print Publication: 2025).Publisher: Public Library of Science Country of Publication: United States NLM ID: 101285081 Publication Model: eCollection Cited Medium: Internet

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Academic Journal

mTORC2 is crucial for regulating the recombinant Mycobacterium tuberculosis CFP-10 protein-induced phagocytosis in macrophages.

  • Authors : Huang XH; The School of Laboratory Medicine & Life Sciences, Key Laboratory of Laboratory Medicine, Wenzhou Medical University, Ministry of Education of China, Wenzhou, Zhejiang, 325035, China.; Wang Y

Subjects: Phagocytosis*/Phagocytosis*/Phagocytosis*/immunology ; Macrophages*/Macrophages*/Macrophages*/immunology ; Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/immunology

  • Source: BMC immunology [BMC Immunol] 2025 May 09; Vol. 26 (1), pp. 36. Date of Electronic Publication: 2025 May 09.Publisher: BioMed Central Country of Publication: England NLM ID: 100966980 Publication Model: Electronic Cited Medium: Internet ISSN: 1471-2172

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Academic Journal

Insights into Active Site Cysteine Residues in Mycobacterium tuberculosis Enzymes: Potential Targets for Anti-Tuberculosis Intervention.

  • Authors : Faponle AS; Department of Biochemistry, Faculty of Basic Medical Sciences, Sagamu Campus, Olabisi Onabanjo University, Ago-Iwoye 120107, Nigeria.; Gauld JW

Subjects: Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/enzymology ; Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/drug effects ; Cysteine*/Cysteine*/Cysteine*/metabolism

  • Source: International journal of molecular sciences [Int J Mol Sci] 2025 Apr 18; Vol. 26 (8). Date of Electronic Publication: 2025 Apr 18.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

Mycobacterium susceptibility to ivermectin by inhibition of eccD3, an ESX-3 secretion system component.

  • Authors : Granados-Tristán AL; Departamento de Biología Molecular, Centro de Investigación Biomédica del Noreste, Instituto Mexicano del Seguro Social, Monterrey, Nuevo León, México.; Facultad de Ciencias Biológicas, Universidad Autónoma de Nuevo León (UANL), San Nicolás de los Garza, Nuevo León, México.

Subjects: Ivermectin*/Ivermectin*/Ivermectin*/pharmacology ; Ivermectin*/Ivermectin*/Ivermectin*/chemistry ; Bacterial Proteins*/Bacterial Proteins*/Bacterial Proteins*/chemistry

  • Source: PLoS computational biology [PLoS Comput Biol] 2025 Apr 17; Vol. 21 (4), pp. e1012936. Date of Electronic Publication: 2025 Apr 17 (Print Publication: 2025).Publisher: Public Library of Science Country of Publication: United States NLM ID: 101238922 Publication Model: eCollection Cited Medium: Internet

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Academic Journal

Single-stranded DNA drives σ subunit loading onto mycobacterial RNA polymerase to unlock initiation-competent conformations.

  • Authors : Vishwakarma RK; Institut de Recherche en Infectiologie de Montpellier, Univ Montpellier, CNRS, Montpellier 34293, France.; Centre de Biologie Structurale, Univ Montpellier, CNRS, INSERM, Montpellier 34090, France.

Subjects: DNA, Single-Stranded*/DNA, Single-Stranded*/DNA, Single-Stranded*/metabolism ; DNA, Single-Stranded*/DNA, Single-Stranded*/DNA, Single-Stranded*/chemistry ; DNA, Single-Stranded*/DNA, Single-Stranded*/DNA, Single-Stranded*/genetics

  • Source: Nucleic acids research [Nucleic Acids Res] 2025 Apr 10; Vol. 53 (7).Publisher: Oxford University Press Country of Publication: England NLM ID: 0411011 Publication Model: Print Cited Medium: Internet ISSN:

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Academic Journal

Early secretory antigen target of 6-kDa of Mycobacterium tuberculosis inhibits macrophage apoptosis and host defense via TLR2.

  • Authors : Zhang L; Anhui Provincial Key Laboratory of Immunology in Chronic Diseases, Anhui Provincial Key Laboratory of Infection and Immunology, and Department of Laboratory Medicine, Bengbu Medical University, Bengbu, Anhui, China.; Yiwu Traditional Chinese Medicine Hospital, Jinhua, Zhejiang, China.

Subjects: Apoptosis*/Apoptosis*/Apoptosis*/physiology ; Apoptosis*/Apoptosis*/Apoptosis*/drug effects ; Apoptosis*/Apoptosis*/Apoptosis*/immunology

  • Source: Respiratory research [Respir Res] 2025 Apr 09; Vol. 26 (1), pp. 131. Date of Electronic Publication: 2025 Apr 09.Publisher: BioMed Central Ltd Country of Publication: England NLM ID: 101090633 Publication Model: Electronic Cited Medium: Internet ISSN:

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Academic Journal

NapR Regulates the Expression of Phosphoserine Aminotransferase SerC to Modulate Biofilm Formation and Resistance to Serine Stress of Mycobacteria.

  • Authors : Guo M; State Key Laboratory for Conservation and Utilization of Subtropical Agro-Bioresources, College of Life Science and Technology, Guangxi University, Nanning 530004, China.; Ling X

Subjects: Biofilms*/Biofilms*/Biofilms*/growth & development ; Serine*/Serine*/Serine*/metabolism ; Gene Expression Regulation, Bacterial*

  • Source: International journal of molecular sciences [Int J Mol Sci] 2025 Feb 28; Vol. 26 (5). Date of Electronic Publication: 2025 Feb 28.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

In situ and in vitro cryo-EM reveal structures of mycobacterial encapsulin assembly intermediates.

  • Authors : Berger C; Division of Nanoscopy, Maastricht Multimodal Molecular Imaging Institute, Maastricht University, Maastricht, The Netherlands. .; Structural Biology, The Rosalind Franklin Institute, Harwell Science & Innovation Campus, Didcot, United Kingdom. .

Subjects: Cryoelectron Microscopy*/Cryoelectron Microscopy*/Cryoelectron Microscopy*/methods ; Bacterial Proteins*/Bacterial Proteins*/Bacterial Proteins*/metabolism ; Bacterial Proteins*/Bacterial Proteins*/Bacterial Proteins*/chemistry

  • Source: Communications biology [Commun Biol] 2025 Feb 15; Vol. 8 (1), pp. 245. Date of Electronic Publication: 2025 Feb 15.Publisher: Nature Publishing Group UK Country of Publication: England NLM ID: 101719179 Publication Model: Electronic Cited Medium: Internet ISSN:

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Academic Journal

Identification of new ClpC1-NTD binders for Mycobacterium tuberculosis drug development.

  • Authors : Weinhäupl K; Institute for Research and Innovation in HealthI3S, Porto, Portugal. .; Meuret L

Subjects: Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/drug effects ; Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/Mycobacterium tuberculosis*/metabolism ; Bacterial Proteins*/Bacterial Proteins*/Bacterial Proteins*/metabolism

  • Source: Scientific reports [Sci Rep] 2025 Feb 03; Vol. 15 (1), pp. 4146. Date of Electronic Publication: 2025 Feb 03.Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101563288 Publication Model: Electronic Cited Medium: Internet ISSN:

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