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  • 1-10 ل  4,098 نتائج ل ""Structure-Activity Relationship""
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Academic Journal

Synthesis and Structure-Activity Relationship (SAR) Studies on New 4-Aminoquinoline-Hydrazones and Isatin Hybrids as Promising Antibacterial Agents.

  • Authors : Ubaid A; Medicinal Chemistry Laboratory, Department of Biosciences, Jamia Millia Islamia, New Delhi 110025, India.; Shakir M

Subjects: Anti-Bacterial Agents*/Anti-Bacterial Agents*/Anti-Bacterial Agents*/pharmacology ; Anti-Bacterial Agents*/Anti-Bacterial Agents*/Anti-Bacterial Agents*/chemistry ; Anti-Bacterial Agents*/Anti-Bacterial Agents*/Anti-Bacterial Agents*/chemical synthesis

  • Source: Molecules (Basel, Switzerland) [Molecules] 2024 Dec 06; Vol. 29 (23). Date of Electronic Publication: 2024 Dec 06.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Development of Naphthalene-Derivative Bis-QACs as Potent Antimicrobials: Unraveling Structure-Activity Relationship and Microbiological Properties.

  • Authors : Frolov NA; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky Prospect 47, 119991 Moscow, Russia.; Seferyan MA

Subjects: Naphthalenes*/Naphthalenes*/Naphthalenes*/pharmacology ; Naphthalenes*/Naphthalenes*/Naphthalenes*/chemistry ; Biofilms*/Biofilms*/Biofilms*/drug effects

  • Source: Molecules (Basel, Switzerland) [Molecules] 2024 Nov 22; Vol. 29 (23). Date of Electronic Publication: 2024 Nov 22.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Targeting bacterial growth in biofilm conditions: rational design of novel inhibitors to mitigate clinical and food contamination using QSAR.

  • Authors : Galvez-Llompart M; Department of Preventive Medicine and Public Health, Food Science, Toxicology and Forensic Medicine, Faculty of Pharmacy, University of Valencia, Burjassot, Spain.; Department of Physical Chemistry, University of Valencia, Burjassot, Spain.

Subjects: Biofilms*/Biofilms*/Biofilms*/drug effects ; Quantitative Structure-Activity Relationship* ; Anti-Bacterial Agents*/Anti-Bacterial Agents*/Anti-Bacterial Agents*/pharmacology

  • Source: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2024 Dec; Vol. 39 (1), pp. 2330907. Date of Electronic Publication: 2024 Apr 23.Publisher: Taylor & Francis Country of Publication: England NLM ID: 101150203 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Evaluation of antibacterial, cytotoxicity, and apoptosis activity of novel chromene-sulfonamide hybrids synthesized under solvent-free conditions and 3D-QSAR modeling studies.

  • Authors : Ghomashi S; Department of Medicinal Chemistry, Shahreza Branch, Islamic Azad University, P.O. Box 311-86145, Shahreza, Isfahan, Iran.; Ghomashi R

Subjects: Quantitative Structure-Activity Relationship* ; Sulfonamides*/Sulfonamides*/Sulfonamides*/chemistry ; Sulfonamides*/Sulfonamides*/Sulfonamides*/pharmacology

  • Source: Scientific reports [Sci Rep] 2024 Jun 05; Vol. 14 (1), pp. 12878. Date of Electronic Publication: 2024 Jun 05.Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101563288 Publication Model: Electronic Cited Medium: Internet ISSN:

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Academic Journal

Design, Synthesis, Antifungal Activity, and 3D-QSAR Study of Novel Quinoxaline-2-Oxyacetate Hydrazide.

  • Authors : Teng P; Jiangsu Key Laboratory of Pesticide Science, College of Sciences, Nanjing Agricultural University, Nanjing 210095, China.; Li Y

Subjects: Quantitative Structure-Activity Relationship* ; Antifungal Agents*/Antifungal Agents*/Antifungal Agents*/pharmacology ; Antifungal Agents*/Antifungal Agents*/Antifungal Agents*/chemical synthesis Rhizoctonia solani; Botrytis cinerea; Alternaria alternata

  • Source: Molecules (Basel, Switzerland) [Molecules] 2024 May 25; Vol. 29 (11). Date of Electronic Publication: 2024 May 25.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Synthesis and antibacterial activity of vanillic acid derivatives containing indole structure.

  • Authors : Zhang J; College of pharmacy, Jiangsu Ocean University. .; Liu Q

Subjects: Anti-Bacterial Agents*/Anti-Bacterial Agents*/Anti-Bacterial Agents*/pharmacology ; Anti-Bacterial Agents*/Anti-Bacterial Agents*/Anti-Bacterial Agents*/chemical synthesis ; Anti-Bacterial Agents*/Anti-Bacterial Agents*/Anti-Bacterial Agents*/chemistry Vibrio harveyi

  • Source: Acta chimica Slovenica [Acta Chim Slov] 2025 Feb 11; Vol. 72 (1), pp. 127-132. Date of Electronic Publication: 2025 Feb 11.Publisher: Slovenian Chemical Society Country of Publication: Slovenia NLM ID: 101247110 Publication Model: Electronic Cited Medium: Internet ISSN:

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Academic Journal

Synthesis and Antimicrobial Activity of 3-Alkylidene-2-Indolone Derivatives.

  • Authors : Huang H; College of Pharmacy, Yanbian University, Yanji 133002, China.; Zhang Y

Subjects: Microbial Sensitivity Tests* ; Anti-Bacterial Agents*/Anti-Bacterial Agents*/Anti-Bacterial Agents*/pharmacology ; Anti-Bacterial Agents*/Anti-Bacterial Agents*/Anti-Bacterial Agents*/chemical synthesis

  • Source: Molecules (Basel, Switzerland) [Molecules] 2024 Nov 15; Vol. 29 (22). Date of Electronic Publication: 2024 Nov 15.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

In vitro and in silico insights into antimicrobial and anticancer activities of novel imidazo[2,1-b][1,3,4]thiadiazoles.

  • Authors : Dwarakanath D; Department of Chemistry, Manipal Institute of Technology, Manipal Academy of Higher Education, Manipal, Karnataka, 576104, India.; Nayak YN

Subjects: Thiadiazoles*/Thiadiazoles*/Thiadiazoles*/chemistry ; Thiadiazoles*/Thiadiazoles*/Thiadiazoles*/pharmacology ; Thiadiazoles*/Thiadiazoles*/Thiadiazoles*/chemical synthesis

  • Source: Scientific reports [Sci Rep] 2024 Dec 30; Vol. 14 (1), pp. 31994. Date of Electronic Publication: 2024 Dec 30.Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101563288 Publication Model: Electronic Cited Medium: Internet ISSN:

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Academic Journal

Elucidation of Antimicrobials and Biofilm Inhibitors Derived from a Polyacetylene Core.

  • Authors : Skeen TL; Department of Chemistry, William & Mary, Williamsburg, VA 23185, USA.; Gresham RL

Subjects: Biofilms*/Biofilms*/Biofilms*/drug effects ; Biofilms*/Biofilms*/Biofilms*/growth & development ; Polyynes*/Polyynes*/Polyynes*/chemistry

  • Source: Molecules (Basel, Switzerland) [Molecules] 2024 Dec 17; Vol. 29 (24). Date of Electronic Publication: 2024 Dec 17.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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  • 1-10 ل  4,098 نتائج ل ""Structure-Activity Relationship""