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Academic Journal

New Insights into the Opioid Analgesic Profile of cis -(-)- N -Normetazocine-derived Ligands.

  • Authors : Costanzo G; Department of Biomedical and Biotechnological Sciences, University of Catania, Via Santa Sofia 97, 95123 Catania, Italy.; Turnaturi R

Subjects: Analgesics, Opioid*/Analgesics, Opioid*/Analgesics, Opioid*/pharmacology ; Receptors, Opioid, mu*/Receptors, Opioid, mu*/Receptors, Opioid, mu*/metabolism; Male

  • Source: Molecules (Basel, Switzerland) [Molecules] 2023 Jun 17; Vol. 28 (12). Date of Electronic Publication: 2023 Jun 17.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

SR-17018 Stimulates Atypical µ-Opioid Receptor Phosphorylation and Dephosphorylation.

  • Authors : Fritzwanker S; Department of Pharmacology and Toxicology, Jena University Hospital, Friedrich Schiller University Jena, Drackendorfer Straße 1, D-07747 Jena, Germany.; Schulz S

Subjects: Analgesics, Opioid*/Analgesics, Opioid*/Analgesics, Opioid*/chemistry ; Analgesics, Opioid*/Analgesics, Opioid*/Analgesics, Opioid*/pharmacology ; Benzimidazoles*/Benzimidazoles*/Benzimidazoles*/chemistry

  • Source: Molecules (Basel, Switzerland) [Molecules] 2021 Jul 27; Vol. 26 (15). Date of Electronic Publication: 2021 Jul 27.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Modulation of the MOP Receptor (μ Opioid Receptor) by Imidazo[1,2- a ]imidazole-5,6-Diones: In Search of the Elucidation of the Mechanism of Action.

  • Authors : Straszak D; Department of Synthesis and Chemical Technology of Pharmaceutical Substances, Faculty of Pharmacy, Medical University, Chodzki 4A, 20-093 Lublin, Poland.; Siwek A

Subjects: Morphine*/Morphine*/Morphine*/pharmacology ; Receptors, Opioid, mu*/Receptors, Opioid, mu*/Receptors, Opioid, mu*/metabolism; Analgesics, Opioid/Analgesics, Opioid/Analgesics, Opioid/therapeutic use

  • Source: Molecules (Basel, Switzerland) [Molecules] 2022 May 04; Vol. 27 (9). Date of Electronic Publication: 2022 May 04.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Modulation of μ-opioid receptor activation by acidic pH is dependent on ligand structure and an ionizable amino acid residue.

  • Authors : Meyer J; Department of Experimental Anesthesiology, Campus Benjamin Franklin, Charité-Universitätsmedizin Berlin, Germany.; Del Vecchio G

Subjects: Enkephalin, Ala(2)-MePhe(4)-Gly(5)-/Enkephalin, Ala(2)-MePhe(4)-Gly(5)-/Enkephalin, Ala(2)-MePhe(4)-Gly(5)-/*pharmacology ; Fentanyl/Fentanyl/Fentanyl/*pharmacology ; Histamine/Histamine/Histamine/*metabolism

  • Source: British journal of pharmacology [Br J Pharmacol] 2019 Dec; Vol. 176 (23), pp. 4510-4520. Date of Electronic Publication: 2019 Dec 05.Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1476-5381

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Academic Journal

Long-term antagonism and allosteric regulation of mu opioid receptors by the novel ligand, methocinnamox.

  • Authors : Zamora JC; Department of Pharmacology, UT Health San Antonio, San Antonio, Texas, USA.; Smith HR

Subjects: Cinnamates/Cinnamates/Cinnamates/*pharmacology ; Morphine Derivatives/Morphine Derivatives/Morphine Derivatives/*pharmacology ; Narcotic Antagonists/Narcotic Antagonists/Narcotic Antagonists/*pharmacology

  • Source: Pharmacology research & perspectives [Pharmacol Res Perspect] 2021 Dec; Vol. 9 (6), pp. e00887.Publisher: John Wiley & Sons Ltd, British Pharmacological Society and American Society for Pharmacology and Experimental Therapeutics Country of Publication: United States

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Academic Journal

Endogenous Opioid Signaling in the Mouse Retina Modulates Pupillary Light Reflex.

  • Authors : Cleymaet AM; Department of Biomedical Sciences, Colorado State University, Ft. Collins, CO 80523, USA.; Department of Clinical Sciences, Colorado State University, Ft. Collins, CO 80523, USA.

Subjects: Opioid Peptides/Opioid Peptides/Opioid Peptides/*genetics ; Receptors, Opioid, mu/Receptors, Opioid, mu/Receptors, Opioid, mu/*genetics ; Retina/Retina/Retina/*metabolism

  • Source: International journal of molecular sciences [Int J Mol Sci] 2021 Jan 08; Vol. 22 (2). Date of Electronic Publication: 2021 Jan 08.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

Positive allosteric modulation of the cannabinoid type-1 receptor (CB1R) in periaqueductal gray (PAG) antagonizes anti-nociceptive and cellular effects of a mu-opioid receptor agonist in morphine-withdrawn rats.

  • Authors : Datta U; Department of Physiology, Louisiana State University Health Science Center, Room 7205 1901 Perdido Street, New Orleans, LA, 70112, USA.; The Jackson Laboratory, Bar Harbor, ME, 04609, USA.

Subjects: Analgesics, Opioid/Analgesics, Opioid/Analgesics, Opioid/*adverse effects ; Morphine/Morphine/Morphine/*adverse effects ; Nociception/Nociception/Nociception/*drug effects

  • Source: Psychopharmacology [Psychopharmacology (Berl)] 2020 Dec; Vol. 237 (12), pp. 3729-3739. Date of Electronic Publication: 2020 Aug 28.Publisher: Springer-Verlag Country of Publication: Germany NLM ID: 7608025 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Voltage modulates the effect of μ-receptor activation in a ligand-dependent manner.

  • Authors : Ruland JG; Department of Pharmacology and Clinical Pharmacy, Philipps-University, Marburg, Germany.; Kirchhofer SB

Subjects: Locus Coeruleus*/Locus Coeruleus*/Locus Coeruleus*/metabolism ; Receptors, Opioid, mu*/Receptors, Opioid, mu*/Receptors, Opioid, mu*/metabolism; Animals

  • Source: British journal of pharmacology [Br J Pharmacol] 2020 Aug; Vol. 177 (15), pp. 3489-3504. Date of Electronic Publication: 2020 May 19.Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1476-5381

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Academic Journal

Activation of μ-opioid receptors by MT-45 (1-cyclohexyl-4-(1,2-diphenylethyl)piperazine) and its fluorinated derivatives.

  • Authors : Baptista-Hon DT; Institute of Academic Anaesthesia, Division of Systems Medicine, School of Medicine, Ninewells Hospital and Medical School, University of Dundee, Dundee, UK.; Smith M

Subjects: Morphine* ; Receptors, Opioid, mu*; Analgesics, Opioid/Analgesics, Opioid/Analgesics, Opioid/pharmacology

  • Source: British journal of pharmacology [Br J Pharmacol] 2020 Aug; Vol. 177 (15), pp. 3436-3448. Date of Electronic Publication: 2020 May 13.Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1476-5381

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Academic Journal

Differential regulation of Cav2.2 channel exon 37 variants by alternatively spliced μ-opioid receptors.

  • Authors : Gandini MA; Department of Physiology and Pharmacology, Alberta Children's Hospital Research Institute, Hotchkiss Brain Institute, Cumming School of Medicine, University of Calgary, Calgary, AB, Canada.; Souza IA

Subjects: Alternative Splicing/Alternative Splicing/Alternative Splicing/*genetics ; Calcium Channels, N-Type/Calcium Channels, N-Type/Calcium Channels, N-Type/*genetics ; Exons/Exons/Exons/*genetics

  • Source: Molecular brain [Mol Brain] 2019 Nov 27; Vol. 12 (1), pp. 98. Date of Electronic Publication: 2019 Nov 27.Publisher: BioMed Central Country of Publication: England NLM ID: 101468876 Publication Model: Electronic Cited Medium: Internet ISSN: 1756-6606

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