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Academic Journal

The Role of Furin and Its Therapeutic Potential in Cardiovascular Disease Risk.

  • Authors : Fry H; Nuffield Department of Population Health, University of Oxford, Oxford OX3 7LF, UK.; Mazidi M

Subjects: Furin*/Furin*/Furin*/metabolism ; Furin*/Furin*/Furin*/genetics ; Cardiovascular Diseases*/Cardiovascular Diseases*/Cardiovascular Diseases*/metabolism

  • Source: International journal of molecular sciences [Int J Mol Sci] 2024 Aug 26; Vol. 25 (17). Date of Electronic Publication: 2024 Aug 26.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

Development and Prospects of Furin Inhibitors for Therapeutic Applications.

Subjects: Furin*/Furin*/Furin*/antagonists & inhibitors ; Furin*/Furin*/Furin*/metabolism; Humans

  • Source: International journal of molecular sciences [Int J Mol Sci] 2024 Aug 24; Vol. 25 (17). Date of Electronic Publication: 2024 Aug 24.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

Screening of Small-Molecule Libraries Using SARS-CoV-2-Derived Sequences Identifies Novel Furin Inhibitors.

  • Authors : Jorkesh A; Department of Pharmaceutical and Pharmacological Science, University of Padova, Via Marzolo, 5, 35131 Padova, Italy.; Department of Biology, University of Padua, Viale G. Colombo 3, 35131 Padova, Italy.

Subjects: Furin*/Furin*/Furin*/antagonists & inhibitors ; Furin*/Furin*/Furin*/metabolism ; SARS-CoV-2*/SARS-CoV-2*/SARS-CoV-2*/drug effects SARS-CoV-2 variants

  • Source: International journal of molecular sciences [Int J Mol Sci] 2024 May 07; Vol. 25 (10). Date of Electronic Publication: 2024 May 07.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

Functional and Multi-Omics Effects of an Optimized CRISPR-Mediated FURIN Depletion in U937 Monocytes.

  • Authors : Chua R; Program in Cardiovascular and Metabolic Disorders, Duke-NUS Medical School, Singapore 169857, Singapore.; Wang L

Subjects: Furin*/Furin*/Furin*/genetics ; Furin*/Furin*/Furin*/metabolism ; Monocytes*/Monocytes*/Monocytes*/metabolism

  • Source: Cells [Cells] 2024 Mar 28; Vol. 13 (7). Date of Electronic Publication: 2024 Mar 28.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101600052 Publication Model: Electronic Cited Medium: Internet ISSN: 2073-4409

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Academic Journal

Vitamin A Status Modulates Epithelial Mesenchymal Transition in the Lung: The Role of Furin.

  • Authors : Cabezuelo MT; Department of Physiology, University of Valencia, 46010 Valencia, Spain.; Centro Salud Safranar, Hospital Universitario Doctor Peset, 46017 Valencia, Spain.

Subjects: Furin*/Furin*/Furin*/metabolism ; Epithelial-Mesenchymal Transition*/Epithelial-Mesenchymal Transition*/Epithelial-Mesenchymal Transition*/drug effects ; Lung*/Lung*/Lung*/metabolism

  • Source: Nutrients [Nutrients] 2024 Apr 15; Vol. 16 (8). Date of Electronic Publication: 2024 Apr 15.Publisher: MDPI Publishing Country of Publication: Switzerland NLM ID: 101521595 Publication Model: Electronic Cited Medium: Internet ISSN:

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Academic Journal

Myelin Basic Protein Attenuates Furin-Mediated Bri2 Cleavage and Postpones Its Membrane Trafficking.

  • Authors : Smirnova EV; Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, 117997 Moscow, Russia.; Timofeev VI

Subjects: Membrane Glycoproteins* ; Furin*/Furin*/Furin*/metabolism; Animals

  • Source: International journal of molecular sciences [Int J Mol Sci] 2024 Feb 23; Vol. 25 (5). Date of Electronic Publication: 2024 Feb 23.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

An Overview of the Role of Furin in Type 2 Diabetes.

  • Authors : Marafie SK; Biochemistry and Molecular Biology Department, Dasman Diabetes Institute, P.O. Box 1180, Dasman 15462, Kuwait.; Al-Mulla F

Subjects: Diabetes Mellitus, Type 2*/Diabetes Mellitus, Type 2*/Diabetes Mellitus, Type 2*/metabolism ; Furin*/Furin*/Furin*/metabolism; Humans

  • Source: Cells [Cells] 2023 Oct 05; Vol. 12 (19). Date of Electronic Publication: 2023 Oct 05.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101600052 Publication Model: Electronic Cited Medium: Internet ISSN: 2073-4409

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Academic Journal

SARS-CoV-2 S Mutations: A Lesson from the Viral World to Understand How Human Furin Works.

  • Authors : Cassari L; Department of Industrial Engineering, University of Padova, Via Marzolo 9, 35131 Padova, Italy.; Pavan A

Subjects: COVID-19* ; Furin*/Furin*/Furin*/metabolism ; SARS-CoV-2*/SARS-CoV-2*/SARS-CoV-2*/genetics

  • Source: International journal of molecular sciences [Int J Mol Sci] 2023 Mar 01; Vol. 24 (5). Date of Electronic Publication: 2023 Mar 01.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

Permethrin as a Potential Furin Inhibitor through a Novel Non-Competitive Allosteric Inhibition.

  • Authors : Feng D; School of Life Science and Biopharmaceutics, Shenyang Pharmaceutical University, 103 Wenhua Road, Shenyang 110016, China.; Ren L

Subjects: Furin*/Furin*/Furin*/antagonists & inhibitors ; Permethrin*/Permethrin*/Permethrin*/pharmacology; Humans

  • Source: Molecules (Basel, Switzerland) [Molecules] 2023 Feb 16; Vol. 28 (4). Date of Electronic Publication: 2023 Feb 16.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Effect of SARS-CoV-2 S protein on the proteolytic cleavage of the epithelial Na+ channel ENaC.

  • Authors : Magaña-Ávila GR; Department of Nephrology and Mineral Metabolism, Instituto Nacional de Ciencias Médicas y Nutrición Salvador Zubirán, Mexico City, Mexico.; Facultad de Medicina, Universidad Nacional Autónoma de México, Mexico City, Mexico.

Subjects: Epithelial Sodium Channels*/Epithelial Sodium Channels*/Epithelial Sodium Channels*/metabolism ; Furin*/Furin*/Furin*/metabolism ; SARS-CoV-2*/SARS-CoV-2*/SARS-CoV-2*/metabolism

  • Source: PloS one [PLoS One] 2024 Apr 25; Vol. 19 (4), pp. e0302436. Date of Electronic Publication: 2024 Apr 25 (Print Publication: 2024).Publisher: Public Library of Science Country of Publication: United States NLM ID: 101285081 Publication Model: eCollection Cited Medium: Internet

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