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Academic Journal

Emerging opportunities of using large language models for translation between drug molecules and indications.

  • Authors : Oniani D; Department of Health Information Management, University of Pittsburgh, Pittsburgh, PA, USA.; Hilsman J

Subjects: Artificial Intelligence* ; Drug Discovery*/Drug Discovery*/Drug Discovery*/methods; Humans

  • Source: Scientific reports [Sci Rep] 2024 May 10; Vol. 14 (1), pp. 10738. Date of Electronic Publication: 2024 May 10.Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101563288 Publication Model: Electronic Cited Medium: Internet ISSN:

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Academic Journal

Elucidating the semantics-topology trade-off for knowledge inference-based pharmacological discovery.

  • Authors : Sosa DN; Stanford University, Department of Biomedical Data Science, Stanford, CA, USA.; Neculae G

Subjects: Semantics* ; Drug Discovery*/Drug Discovery*/Drug Discovery*/methods; Drug Repositioning/Drug Repositioning/Drug Repositioning/methods

  • Source: Journal of biomedical semantics [J Biomed Semantics] 2024 May 01; Vol. 15 (1), pp. 5. Date of Electronic Publication: 2024 May 01.Publisher: Biomed Central Country of Publication: England NLM ID: 101531992 Publication Model: Electronic Cited Medium: Internet ISSN: 2041-1480

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Academic Journal

Connective Tissue Growth Factor: Regulation, Diseases, and Drug Discovery.

  • Authors : Ren M; Key Laboratory of Animal Diseases and Human Health of Sichuan Province, College of Veterinary Medicine, Sichuan Agricultural University, Chengdu 611130, China.; Law Sau Fai Institute for Advancing Translational Medicine in Bone and Joint Diseases (TMBJ), School of Chinese Medicine, Hong Kong Baptist University, Hong Kong SAR, China.

Subjects: Connective Tissue Growth Factor*/Connective Tissue Growth Factor*/Connective Tissue Growth Factor*/metabolism ; Drug Discovery*/Drug Discovery*/Drug Discovery*/methods; Humans

  • Source: International journal of molecular sciences [Int J Mol Sci] 2024 Apr 25; Vol. 25 (9). Date of Electronic Publication: 2024 Apr 25.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

The prospects of automation in drug discovery research using silkworms.

Subjects: Automation, Laboratory* ; Bombyx* ; Drug Discovery*/Drug Discovery*/Drug Discovery*/methods

  • Source: Drug discoveries & therapeutics [Drug Discov Ther] 2024 Jun 06; Vol. 18 (2), pp. 130-133. Date of Electronic Publication: Publisher: Shandong University China-Japan Cooperation Center for Drug Discovery & Screen Country of Publication: Japan NLM ID:

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Academic Journal

Precision cut lung slices: an integrated ex vivo model for studying lung physiology, pharmacology, disease pathogenesis and drug discovery.

  • Authors : Koziol-White C; Rutgers Institute for Translational Medicine and Science, The State University of NJ, 08901, Rutgers, New Brunswick, NJ, USA. .; Gebski E

Subjects: Lung*/Lung*/Lung*/drug effects ; Lung*/Lung*/Lung*/physiopathology ; Lung Diseases*/Lung Diseases*/Lung Diseases*/physiopathology

  • Source: Respiratory research [Respir Res] 2024 Jun 01; Vol. 25 (1), pp. 231. Date of Electronic Publication: 2024 Jun 01.Publisher: BioMed Central Ltd Country of Publication: England NLM ID: 101090633 Publication Model: Electronic Cited Medium: Internet ISSN:

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Academic Journal

D R e A mocracy: A Method to Capitalise on Prior Drug Discovery Efforts to Highlight Candidate Drugs for Repurposing.

  • Authors : Savva K; Bioinformatics Department, The Cyprus Institute of Neurology and Genetics, Nicosia 2370, Cyprus.; Zachariou M

Subjects: Drug Repositioning*/Drug Repositioning*/Drug Repositioning*/methods ; Drug Discovery*/Drug Discovery*/Drug Discovery*/methods; Humans

  • Source: International journal of molecular sciences [Int J Mol Sci] 2024 May 13; Vol. 25 (10). Date of Electronic Publication: 2024 May 13.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

DCGAN-DTA: Predicting drug-target binding affinity with deep convolutional generative adversarial networks.

  • Authors : Kalemati M; Department of Computer Engineering, Sharif University of Technology, Tehran, Iran.; Zamani Emani M

Subjects: Drug Discovery*/Drug Discovery*/Drug Discovery*/methods; Computational Biology/Computational Biology/Computational Biology/methods ; Humans

  • Source: BMC genomics [BMC Genomics] 2024 May 09; Vol. 25 (1), pp. 411. Date of Electronic Publication: 2024 May 09.Publisher: BioMed Central Country of Publication: England NLM ID: 100965258 Publication Model: Electronic Cited Medium: Internet ISSN: 1471-2164

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Academic Journal

Machine learning framework to predict pharmacokinetic profile of small molecule drugs based on chemical structure.

  • Authors : Pillai N; Global DMPK Modeling & Simulation, Sanofi, Cambridge, Massachusetts, USA.; Abos A

Subjects: Machine Learning* ; Drug Discovery*/Drug Discovery*/Drug Discovery*/methods; Animals

  • Source: Clinical and translational science [Clin Transl Sci] 2024 May; Vol. 17 (5), pp. e13824.Publisher: WileyBlackwell Pub Country of Publication: United States NLM ID: 101474067 Publication Model: Print Cited Medium: Internet ISSN:

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Academic Journal

Recent advances in the discovery and development of drugs targeting the kallikrein-kinin system.

  • Authors : Wisniewski P; Individualized Pharmacotherapy, Institute of Pharmaceutical and Medicinal Chemistry, University of Münster, Corrensstr. 48, 48149, Münster, Germany.; Gangnus T

Subjects: Kallikrein-Kinin System*/Kallikrein-Kinin System*/Kallikrein-Kinin System*/physiology ; Drug Discovery*; Humans

  • Source: Journal of translational medicine [J Transl Med] 2024 Apr 26; Vol. 22 (1), pp. 388. Date of Electronic Publication: 2024 Apr 26.Publisher: BioMed Central Country of Publication: England NLM ID: 101190741 Publication Model: Electronic Cited Medium: Internet ISSN: 1479-5876

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Academic Journal

Large-scale chemoproteomics expedites ligand discovery and predicts ligand behavior in cells.

  • Authors : Offensperger F; CeMM, Research Center for Molecular Medicine of the Austrian Academy of Sciences, 1090 Vienna, Austria.; Tin G

Subjects: Drug Discovery* ; Machine Learning* ; Proteomics*/Proteomics*/Proteomics*/methods

  • Source: Science (New York, N.Y.) [Science] 2024 Apr 26; Vol. 384 (6694), pp. eadk5864. Date of Electronic Publication: 2024 Apr 26.Publisher: American Association for the Advancement of Science Country of Publication: United States NLM ID: 0404511 Publication Model: Print-Electronic

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