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Academic Journal

A new method for detection of tumor driver-dependent changes of protein sialylation in a colon cancer cell line reveals nectin-3 as TGFBR2 target.

  • Authors : Lee J; Department of Applied Tumor Biology, Institute of Pathology, University Hospital Heidelberg, Heidelberg, Germany.; Department of Cancer Early Detection, German Cancer Research Center (DKFZ), Heidelberg, Germany.

Subjects: Biochemistry/Biochemistry/Biochemistry/*methods ; Cell Adhesion Molecules/Cell Adhesion Molecules/Cell Adhesion Molecules/*metabolism ; Colonic Neoplasms/Colonic Neoplasms/Colonic Neoplasms/*physiopathology

  • Source: Protein science : a publication of the Protein Society [Protein Sci] 2015 Oct; Vol. 24 (10), pp. 1686-94. Date of Electronic Publication: 2015 Jul 30.Publisher: Cold Spring Harbor Laboratory Press Country of Publication: United States NLM ID: 9211750 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

Comparison of intestinal metabolism of CYP3A substrates between rats and humans: application of portal-systemic concentration difference method.

  • Authors : Kadono K; Analysis and Pharmacokinetics Research Laboratories, Astellas Pharma Inc. , Ibaraki , Japan.; Koakutsu A

Subjects: Biochemistry/Biochemistry/Biochemistry/*methods ; Cytochrome P-450 CYP3A/Cytochrome P-450 CYP3A/Cytochrome P-450 CYP3A/*metabolism ; Intestinal Mucosa/Intestinal Mucosa/Intestinal Mucosa/*metabolism

  • Source: Xenobiotica; the fate of foreign compounds in biological systems [Xenobiotica] 2014 Jun; Vol. 44 (6), pp. 511-21. Date of Electronic Publication: 2013 Dec 12.Publisher: Informa Healthcare Country of Publication: England NLM ID: 1306665 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Method for predicting human intestinal first-pass metabolism of UGT substrate compounds.

  • Authors : Furukawa T; Analysis and Pharmacokinetics Research Laboratories, Astellas Pharma Inc., Ibaraki, Japan. ; Yamano K

Subjects: Biochemistry/Biochemistry/Biochemistry/*methods ; Glucuronides/Glucuronides/Glucuronides/*metabolism ; Glucuronosyltransferase/Glucuronosyltransferase/Glucuronosyltransferase/*metabolism

  • Source: Xenobiotica; the fate of foreign compounds in biological systems [Xenobiotica] 2012 Oct; Vol. 42 (10), pp. 980-8. Date of Electronic Publication: 2012 Apr 27.Publisher: Informa Healthcare Country of Publication: England NLM ID: 1306665 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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