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Academic Journal

Use of a small molecule microarray screen to identify inhibitors of the catalytic RNA subunit of Methanobrevibacter smithii RNase P.

  • Authors : Sidharthan V; Department of Chemistry and Biochemistry, The Ohio State University, Columbus, OH 43210, USA.; Center for RNA Biology, The Ohio State University, Columbus, OH 43210, USA.

Subjects: Ribonuclease P*/Ribonuclease P*/Ribonuclease P*/metabolism ; Ribonuclease P*/Ribonuclease P*/Ribonuclease P*/antagonists & inhibitors ; Ribonuclease P*/Ribonuclease P*/Ribonuclease P*/chemistry

  • Source: Nucleic acids research [Nucleic Acids Res] 2025 Jan 07; Vol. 53 (1).Publisher: Oxford University Press Country of Publication: England NLM ID: 0411011 Publication Model: Print Cited Medium:

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Academic Journal

Structure-based discovery of first inhibitors targeting the helicase activity of human PIF1.

  • Authors : Wever MJA; Edelris, Bioparc, Bioserra 1 Building, 69008 Lyon, France.; Univ. Grenoble Alpes, CNRS, DCM, 38000 Grenoble, France.

Subjects: DNA Helicases*/DNA Helicases*/DNA Helicases*/metabolism ; DNA Helicases*/DNA Helicases*/DNA Helicases*/antagonists & inhibitors ; DNA Helicases*/DNA Helicases*/DNA Helicases*/chemistry

  • Source: Nucleic acids research [Nucleic Acids Res] 2024 Nov 11; Vol. 52 (20), pp. 12616-12632.Publisher: Oxford University Press Country of Publication: England NLM ID: 0411011 Publication Model: Print Cited Medium:

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Academic Journal

Janus Kinase Inhibitors Differentially Inhibit Specific Cytokine Signals in the Mesenteric Lymph Node Cells of Inflammatory Bowel Disease Patients.

Subjects: Janus Kinase Inhibitors*/Janus Kinase Inhibitors*/Janus Kinase Inhibitors*/pharmacology ; Janus Kinase Inhibitors*/Janus Kinase Inhibitors*/Janus Kinase Inhibitors*/therapeutic use ; Piperidines*/Piperidines*/Piperidines*/pharmacology

  • Source: Journal of Crohn's & colitis [J Crohns Colitis] 2024 Apr 23; Vol. 18 (4), pp. 628-637.Publisher: Oxford University Press Country of Publication: England NLM ID: 101318676 Publication Model: Print Cited Medium:

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Academic Journal

PARP1-TRIM44-MRN loop dictates the response to PARP inhibitors.

  • Authors : Kim Y; Department of Biochemistry, Ajou University School of Medicine, Suwon 16499, Republic of Korea.; Min S

Subjects: Poly(ADP-ribose) Polymerase Inhibitors*/Poly(ADP-ribose) Polymerase Inhibitors*/Poly(ADP-ribose) Polymerase Inhibitors*/pharmacology ; Poly (ADP-Ribose) Polymerase-1*/Poly (ADP-Ribose) Polymerase-1*/Poly (ADP-Ribose) Polymerase-1*/metabolism ; Poly (ADP-Ribose) Polymerase-1*/Poly (ADP-Ribose) Polymerase-1*/Poly (ADP-Ribose) Polymerase-1*/genetics

  • Source: Nucleic acids research [Nucleic Acids Res] 2024 Oct 28; Vol. 52 (19), pp. 11720-11737.Publisher: Oxford University Press Country of Publication: England NLM ID: 0411011 Publication Model: Print Cited Medium:

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Academic Journal

Single-molecule studies reveal the off-pathway early paused state intermediates as a target of streptolydigin inhibition of RNA polymerase and its dramatic enhancement by Gre factors.

  • Authors : Arseniev A; Peter the Great St. Petersburg Polytechnic University, Research Center of Nanobiotechnologies, Polytechnicheskaya, 29 B, Saint Petersburg, 195251,Russia.; Institute of Molecular Genetics, Russian Academy of Sciences, Kurchatov Sq., 2, Moscow, 123182, Russia.

Subjects: DNA-Directed RNA Polymerases*/DNA-Directed RNA Polymerases*/DNA-Directed RNA Polymerases*/metabolism ; DNA-Directed RNA Polymerases*/DNA-Directed RNA Polymerases*/DNA-Directed RNA Polymerases*/chemistry ; DNA-Directed RNA Polymerases*/DNA-Directed RNA Polymerases*/DNA-Directed RNA Polymerases*/antagonists & inhibitors

  • Source: Nucleic acids research [Nucleic Acids Res] 2025 Jan 07; Vol. 53 (1).Publisher: Oxford University Press Country of Publication: England NLM ID: 0411011 Publication Model: Print Cited Medium:

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Academic Journal

Treatment of Antibiotic Refractory Chronic Pouchitis With JAK Inhibitors and S1P Receptor Modulators: An ECCO CONFER Multicentre Case Series.

  • Authors : Ribaldone DG; Department of Medical Sciences, Division of Gastroenterology, University of Turin, Turin, Italy.; Testa G

Subjects: Pouchitis*/Pouchitis*/Pouchitis*/drug therapy ; Janus Kinase Inhibitors*/Janus Kinase Inhibitors*/Janus Kinase Inhibitors*/therapeutic use ; Anti-Bacterial Agents*/Anti-Bacterial Agents*/Anti-Bacterial Agents*/therapeutic use

  • Source: Journal of Crohn's & colitis [J Crohns Colitis] 2024 May 31; Vol. 18 (5), pp. 720-726.Publisher: Oxford University Press Country of Publication: England NLM ID: 101318676 Publication Model: Print Cited Medium:

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Academic Journal

Emerging role of topical Janus kinase inhibitors in dermatological disorders: a review.

  • Authors : Dogra S; Department of Dermatology, Venereology and Leprology, Postgraduate Institute of Medical Education and Research, Chandigarh, India.; Sharma A

Subjects: Janus Kinase Inhibitors*/Janus Kinase Inhibitors*/Janus Kinase Inhibitors*/therapeutic use ; Dermatitis, Atopic*/Dermatitis, Atopic*/Dermatitis, Atopic*/drug therapy ; Vitiligo*

  • Source: Clinical and experimental dermatology [Clin Exp Dermatol] 2023 Sep 19; Vol. 48 (10), pp. 1102-1112.Publisher: Oxford University Press Country of Publication: England NLM ID: 7606847 Publication Model: Print Cited Medium:

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