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Academic Journal

Exploring Amantadine Derivatives as Urease Inhibitors: Molecular Docking and Structure-Activity Relationship (SAR) Studies.

  • Authors : Ahmed A; Department of Chemistry, Quaid-I-Azam University, Islamabad 45320, Pakistan.; Saeed A

Subjects: Structure-Activity Relationship*; Enzyme Inhibitors/Enzyme Inhibitors/Enzyme Inhibitors/*chemistry ; Helicobacter Infections/Helicobacter Infections/Helicobacter Infections/*drug therapy

  • Source: Molecules (Basel, Switzerland) [Molecules] 2021 Nov 25; Vol. 26 (23). Date of Electronic Publication: 2021 Nov 25.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium:

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Academic Journal

The Enigmatic Metallothioneins: A Case of Upward-Looking Research.

  • Authors : Abdin AY; Division of Bioorganic Chemistry, School of Pharmacy, Saarland University, D-66123 Saarbruecken, Germany.; Univ. Lille, CNRS, Centrale Lille, Univ. Artois, UMR 8181-UCCS-Unité de Catalyse et Chimie du Solide, F-59000 Lille, France.

Subjects: Structure-Activity Relationship*; Metallothionein/Metallothionein/Metallothionein/*genetics ; Mollusca/Mollusca/Mollusca/*genetics

  • Source: International journal of molecular sciences [Int J Mol Sci] 2021 Jun 01; Vol. 22 (11). Date of Electronic Publication: 2021 Jun 01.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium:

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Academic Journal

Effects of Modifications on the Immunosuppressive Properties of Cyclolinopeptide A and Its Analogs in Animal Experimental Models.

  • Authors : Zimecki M; Laboratory of Immunobiology, Hirszfeld Institute of Immunology and Experimental Therapy, Polish Academy of Sciences, R. Weigla Str. 12, 53-114 Wrocław, Poland.; Kaczmarek K

Subjects: Structure-Activity Relationship*; Amino Acid Sequence/Amino Acid Sequence/Amino Acid Sequence/*genetics ; Peptides/Peptides/Peptides/*genetics

  • Source: Molecules (Basel, Switzerland) [Molecules] 2021 Apr 27; Vol. 26 (9). Date of Electronic Publication: 2021 Apr 27.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium:

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Academic Journal

Probing the Structure and Function of the Cytosolic Domain of the Human Zinc Transporter ZnT8 with Nickel(II) Ions.

  • Authors : Catapano MC; Departments of Biochemistry and Nutritional Sciences, School of Life Course Sciences, Faculty of Life Sciences and Medicine, King's College London, Franklin-Wilkins Bldg, 150 Stamford St., London SE1 9NH, UK.; Department of Analytical Chemistry, Faculty of Pharmacy in Hradec Králové, Charles University, Heyrovského 1203, 500 05 Hradec Králové, Czech Republic.

Subjects: Structure-Activity Relationship*; Carrier Proteins/Carrier Proteins/Carrier Proteins/*ultrastructure ; Insulin/Insulin/Insulin/*genetics

  • Source: International journal of molecular sciences [Int J Mol Sci] 2021 Mar 14; Vol. 22 (6). Date of Electronic Publication: 2021 Mar 14.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium:

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Academic Journal

Structure-Function Relationship Study of a Secretory Amoebic Phosphatase: A Computational-Experimental Approach.

  • Authors : Terán-Ramírez C; Biotechnology and Biosciences Research Group, Faculty of Chemical Sciences and Engineering, Autonomous University of Baja California, Tijuana 22390, Mexico.; Mares-Alejandre RE

Subjects: Structure-Activity Relationship*; Entamoeba histolytica/Entamoeba histolytica/Entamoeba histolytica/*enzymology ; Phosphoric Monoester Hydrolases/Phosphoric Monoester Hydrolases/Phosphoric Monoester Hydrolases/*chemistry

  • Source: International journal of molecular sciences [Int J Mol Sci] 2021 Feb 22; Vol. 22 (4). Date of Electronic Publication: 2021 Feb 22.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium:

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Academic Journal

An Investigation of Structure-Activity Relationships of Azolylacryloyl Derivatives Yielded Potent and Long-Acting Hemoglobin Modulators for Reversing Erythrocyte Sickling.

  • Authors : Omar AM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, King Abdulaziz University, Alsulaymanyah, Jeddah 21589, Saudi Arabia.; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Al-Azhar University, Cairo 11884, Egypt.

Subjects: Structure-Activity Relationship*; Anemia, Sickle Cell/Anemia, Sickle Cell/Anemia, Sickle Cell/*drug therapy ; Hemoglobins/Hemoglobins/Hemoglobins/*genetics

  • Source: Biomolecules [Biomolecules] 2020 Nov 02; Vol. 10 (11). Date of Electronic Publication: 2020 Nov 02.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101596414 Publication Model: Electronic Cited Medium:

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Academic Journal

Importance of Fluorine in Benzazole Compounds.

  • Authors : Al-Harthy T; Department of Basic Sciences, College of Applied and Health Sciences, A'Sharqiyah University, Ibra 400, Oman.; Zoghaib W

Subjects: Structure-Activity Relationship*; Benzimidazoles/Benzimidazoles/Benzimidazoles/*chemistry ; Benzothiazoles/Benzothiazoles/Benzothiazoles/*chemistry

  • Source: Molecules (Basel, Switzerland) [Molecules] 2020 Oct 14; Vol. 25 (20). Date of Electronic Publication: 2020 Oct 14.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium:

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Academic Journal

Computational Method for Quantitative Comparison of Activity Landscapes on the Basis of Image Data.

  • Authors : Iqbal J; Department of Life Science Informatics, B-IT, LIMES Program Unit Chemical Biology and Medicinal Chemistry, Rheinische Friedrich-Wilhelms-Universität, Endenicher Allee 19c, D-53115 Bonn, Germany.; Vogt M

Subjects: Drug Design* ; Drug Discovery* ; Machine Learning*

  • Source: Molecules (Basel, Switzerland) [Molecules] 2020 Aug 29; Vol. 25 (17). Date of Electronic Publication: 2020 Aug 29.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium:

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Academic Journal

Antiplasmodial Activity, Cytotoxicity and Structure-Activity Relationship Study of Cyclopeptide Alkaloids.

  • Authors : Tuenter E; Natural Products & Food Research and Analysis (NatuRA), Department of Pharmaceutical Sciences, University of Antwerp, Universiteitsplein 1, 2610 Antwerp, Belgium. .; Segers K

Subjects: Structure-Activity Relationship*; Alkaloids/Alkaloids/Alkaloids/*chemistry ; Alkaloids/Alkaloids/Alkaloids/*pharmacology

  • Source: Molecules (Basel, Switzerland) [Molecules] 2017 Feb 02; Vol. 22 (2). Date of Electronic Publication: 2017 Feb 02.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium:

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Academic Journal

Molecular Structure, Binding Affinity, and Biological Activity in the Epigenome.

  • Authors : Zsidó BZ; Department of Pharmacology and Pharmacotherapy, Medical School, University of Pécs, Szigeti út 12, 7624 Pécs, Hungary.; Hetényi C

Subjects: Epigenome* ; Structure-Activity Relationship*; DNA/DNA/DNA/*chemistry

  • Source: International journal of molecular sciences [Int J Mol Sci] 2020 Jun 10; Vol. 21 (11). Date of Electronic Publication: 2020 Jun 10.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium:

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