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Academic Journal

Rosuvastatin blocks hERG current and prolongs cardiac repolarization.

  • Authors : Plante I; CRCHUM, Research Center, Centre Hospitalier de l'Université de Montréal, Montreal, Quebec, Canada H2W 1T7.; Vigneault P

Subjects: Fluorobenzenes/Fluorobenzenes/Fluorobenzenes/*pharmacology ; Heart/Heart/Heart/*drug effects ; Hydroxymethylglutaryl-CoA Reductase Inhibitors/Hydroxymethylglutaryl-CoA Reductase Inhibitors/Hydroxymethylglutaryl-CoA Reductase Inhibitors/*pharmacology

  • Source: Journal of pharmaceutical sciences [J Pharm Sci] 2012 Feb; Vol. 101 (2), pp. 868-78. Date of Electronic Publication: 2011 Nov 11.Publisher: Elsevier Country of Publication: United States NLM ID: 2985195R Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

The Use of Transporter Probe Drug Cocktails for the Assessment of Transporter-Based Drug-Drug Interactions in a Clinical Setting-Proposal of a Four Component Transporter Cocktail.

  • Authors : Ebner T; Department of Drug Metabolism and Pharmacokinetics, Boehringer Ingelheim Pharma GmbH and Co. KG, Biberach, Germany.; Ishiguro N

Subjects: ATP-Binding Cassette Transporters/ATP-Binding Cassette Transporters/ATP-Binding Cassette Transporters/*metabolism ; Digoxin/Digoxin/Digoxin/*metabolism ; Furosemide/Furosemide/Furosemide/*metabolism

  • Source: Journal of pharmaceutical sciences [J Pharm Sci] 2015 Sep; Vol. 104 (9), pp. 3220-8. Date of Electronic Publication: 2015 May 15.Publisher: Elsevier Country of Publication: United States NLM ID: 2985195R Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Involvement of PtdIns(4,5)P2 in the regulatory mechanism of small intestinal P-glycoprotein expression.

  • Authors : Kobori T; Department of Clinical Pharmacy, School of Pharmaceutical Sciences, Kobe Gakuin University, Kobe, Japan.; Harada S

Subjects: ATP Binding Cassette Transporter, Subfamily B/ATP Binding Cassette Transporter, Subfamily B/ATP Binding Cassette Transporter, Subfamily B/*biosynthesis ; Intestine, Small/Intestine, Small/Intestine, Small/*metabolism ; Phosphatidylinositol 4,5-Diphosphate/Phosphatidylinositol 4,5-Diphosphate/Phosphatidylinositol 4,5-Diphosphate/*physiology

  • Source: Journal of pharmaceutical sciences [J Pharm Sci] 2014 Feb; Vol. 103 (2), pp. 743-51. Date of Electronic Publication: 2013 Dec 05.Publisher: Elsevier Country of Publication: United States NLM ID: 2985195R Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Activation of ERM-family proteins via RhoA-ROCK signaling increases intestinal P-gp expression and leads to attenuation of oral morphine analgesia.

  • Authors : Kobori T; Department of Clinical Pharmacy, School of Pharmaceutical Sciences, Kobe Gakuin University, Chuo-ku, Kobe 650-8586, Japan.; Harada S

Subjects: ATP Binding Cassette Transporter, Subfamily B, Member 1/ATP Binding Cassette Transporter, Subfamily B, Member 1/ATP Binding Cassette Transporter, Subfamily B, Member 1/*metabolism ; Analgesics, Opioid/Analgesics, Opioid/Analgesics, Opioid/*therapeutic use ; Antineoplastic Agents, Phytogenic/Antineoplastic Agents, Phytogenic/Antineoplastic Agents, Phytogenic/*therapeutic use

  • Source: Journal of pharmaceutical sciences [J Pharm Sci] 2013 Mar; Vol. 102 (3), pp. 1095-105. Date of Electronic Publication: 2013 Jan 09.Publisher: Elsevier Country of Publication: United States NLM ID: 2985195R Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Improved pharmacokinetic and bioavailability support of drug discovery using serial blood sampling in mice.

  • Authors : Peng SX; Johnson & Johnson Pharmaceutical Research & Development, Welsh & McKean Roads, Spring House, Pennsylvania 19477, USA. ; Rockafellow BA

Subjects: Biological Availability* ; Pharmacokinetics*; Pharmaceutical Preparations/Pharmaceutical Preparations/Pharmaceutical Preparations/*metabolism

  • Source: Journal of pharmaceutical sciences [J Pharm Sci] 2009 May; Vol. 98 (5), pp. 1877-84.Publisher: Elsevier Country of Publication: United States NLM ID: 2985195R Publication Model: Print Cited Medium: Internet ISSN: 1520-6017

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