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  • 1-10 ل  2,635 نتائج ل ""Structure-activity""

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Publication : journal of enzyme inhibition and medicinal chemistry
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Academic Journal

Discovery of natural anthraquinones as potent inhibitors against pancreatic lipase: structure-activity relationships and inhibitory mechanism

Subjects: Pancreatic lipase; inhibitor; structure-activity relationships

  • Source: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 39, Iss 1 (2024)

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Academic Journal

Structure-activity exploration of a small-molecule allosteric inhibitor of T790M/L858R double mutant EGFR.

  • Authors : Foschi F; Department of Life Sciences, University of Modena and Reggio Emilia, Modena, Italy.; Department of Chemistry, University of Milano, Milano, Italy.

Subjects: Lung Neoplasms*/Lung Neoplasms*/Lung Neoplasms*/drug therapy ; Lung Neoplasms*/Lung Neoplasms*/Lung Neoplasms*/genetics ; Lung Neoplasms*/Lung Neoplasms*/Lung Neoplasms*/metabolism

  • Source: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2023 Dec; Vol. 38 (1), pp. 239-245.Publisher: Taylor & Francis Country of Publication: England NLM ID: 101150203 Publication Model: Print Cited Medium: Internet ISSN: 1475-6374

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Academic Journal

Curcumin analogues exert potent inhibition on human and rat gonadal 3β-hydroxysteroid dehydrogenases as potential therapeutic agents: structure-activity relationship and in silico docking.

  • Authors : Qiao X; Department of Anesthesiology and Perioperative Medicine, the Second Affiliated Hospital and Yuying Children's Hospital of Wenzhou Medical University, Wenzhou, China.; Ye L

Subjects: Curcumin*/Curcumin*/Curcumin*/pharmacology; Humans ; Rats

  • Source: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2023 Dec; Vol. 38 (1), pp. 2205052.Publisher: Taylor & Francis Country of Publication: England NLM ID: 101150203 Publication Model: Print Cited Medium: Internet ISSN: 1475-6374

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Academic Journal

Synthesis and structure-activity relationships of pyrazole-based inhibitors of meprin α and β.

  • Authors : Tan K; Department of Drug Design and Target Validation MWT, Fraunhofer Institute for Cell Therapy and Immunology IZI, Biocenter, Halle (Saale), Germany.; Jäger C

Subjects: Metalloendopeptidases* ; Metalloproteases*/Metalloproteases*/Metalloproteases*/metabolism; Structure-Activity Relationship

  • Source: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2023 Dec; Vol. 38 (1), pp. 2165648.Publisher: Taylor & Francis Country of Publication: England NLM ID: 101150203 Publication Model: Print Cited Medium: Internet ISSN: 1475-6374

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Academic Journal

Structure-activity exploration of a small-molecule allosteric inhibitor of T790M/L858R double mutant EGFR

Subjects: EGFR inhibitors; allosteric inhibitors; anticancer drugs

  • Source: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1, Pp 239-245 (2023)

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Academic Journal

Paving the way towards effective plant-based inhibitors of hyaluronidase and tyrosinase: a critical review on a structure–activity relationship

Subjects: Hyaluronidase; tyrosinase plant-based inhibitors; structure–activity relationship

  • Source: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 37, Iss 1, Pp 1120-1195 (2022)

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Academic Journal

Curcumin analogues exert potent inhibition on human and rat gonadal 3β-hydroxysteroid dehydrogenases as potential therapeutic agents: structure-activity relationship and in silico docking

Subjects: Curcumin analogues; gonad 3β-HSD; curcumin metabolite

  • Source: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1 (2023)

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Academic Journal

Synthesis and structure–activity relationships of pyrazole-based inhibitors of meprin α and β

Subjects: Meprin; metalloprotease; hydroxamate

  • Source: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1 (2023)

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Academic Journal

Paving the way towards effective plant-based inhibitors of hyaluronidase and tyrosinase: a critical review on a structure-activity relationship.

  • Authors : Gębalski J; Department of Pharmaceutical Botany and Pharmacognosy, Ludwik Rydygier Collegium Medicum, Nicolaus Copernicus University, Bydgoszcz, Poland.; Graczyk F

Subjects: Hyaluronoglucosaminidase*/Hyaluronoglucosaminidase*/Hyaluronoglucosaminidase*/metabolism ; Monophenol Monooxygenase*; Enzyme Inhibitors/Enzyme Inhibitors/Enzyme Inhibitors/chemistry

  • Source: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2022 Dec; Vol. 37 (1), pp. 1120-1195.Publisher: Taylor & Francis Country of Publication: England NLM ID: 101150203 Publication Model: Print Cited Medium: Internet ISSN: 1475-6374

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Academic Journal

Synthesis and preliminary structure-activity relationship study of 3-methylquinazolinone derivatives as EGFR inhibitors with enhanced antiproliferative activities against tumour cells

Subjects: quinazolinone; egfr; kinase inhibitor

  • Source: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 36, Iss 1, Pp 1205-1216 (2021)

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  • 1-10 ل  2,635 نتائج ل ""Structure-activity""