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Academic Journal

The mechanism of non-blocking inhibition of sodium channels revealed by conformation-selective photolabeling.

  • Authors : Földi MC; MTA-ELTE NAP B Opto-Neuropharmacology Group, Budapest, Hungary.; Plant Protection Institute, Centre for Agricultural Research, Martonvásár, Hungary.

Subjects: Sodium Channel Blockers*/Sodium Channel Blockers*/Sodium Channel Blockers*/pharmacology ; Sodium Channels*/Sodium Channels*/Sodium Channels*/metabolism; Binding Sites

  • Source: British journal of pharmacology [Br J Pharmacol] 2021 Mar; Vol. 178 (5), pp. 1200-1217. Date of Electronic Publication: 2021 Feb 01.Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1476-5381

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Academic Journal

Riluzole protects against cardiac ischaemia and reperfusion damage via block of the persistent sodium current.

  • Authors : Weiss S; The John Curtin School of Medical Research, The Australian National University, Canberra, ACT, Australia.; Benoist D

Subjects: Myocardial Reperfusion Injury/Myocardial Reperfusion Injury/Myocardial Reperfusion Injury/*prevention & control ; Riluzole/Riluzole/Riluzole/*pharmacology ; Sodium Channels/Sodium Channels/Sodium Channels/*drug effects

  • Source: British journal of pharmacology [Br J Pharmacol] 2010 Jul; Vol. 160 (5), pp. 1072-82.Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print Cited Medium: Internet ISSN: 1476-5381 (Electronic)

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Academic Journal

Riluzole activates TRPC5 channels independently of PLC activity.

  • Authors : Richter JM; Rudolf-Boehm-Institute of Pharmacology and Toxicology, University of Leipzig, Leipzig, Germany.; Schaefer M

Subjects: Ion Channel Gating/Ion Channel Gating/Ion Channel Gating/*drug effects ; Riluzole/Riluzole/Riluzole/*pharmacology ; TRPC Cation Channels/TRPC Cation Channels/TRPC Cation Channels/*agonists

  • Source: British journal of pharmacology [Br J Pharmacol] 2014 Jan; Vol. 171 (1), pp. 158-70.Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print Cited Medium: Internet ISSN: 1476-5381 (Electronic)

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Academic Journal

The beta-lactam antibiotic, ceftriaxone, attenuates morphine-evoked hyperthermia in rats.

  • Authors : Rawls SM; Department of Pharmaceutical Sciences, Temple University School of Pharmacy, Philadelphia, PA 19140, USA. ; Tallarida R

Subjects: Ceftriaxone/Ceftriaxone/Ceftriaxone/*pharmacology ; Fever/Fever/Fever/*prevention & control ; Morphine/Morphine/Morphine/*toxicity

  • Source: British journal of pharmacology [Br J Pharmacol] 2007 Aug; Vol. 151 (7), pp. 1095-102. Date of Electronic Publication: 2007 Jun 25.Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print-Electronic Cited Medium: Print ISSN: 0007-1188 (Print)

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Academic Journal

Riluzole inhibits spontaneous Ca2+ signaling in neuroendocrine cells by activation of K+ channels and inhibition of Na+ channels.

  • Authors : Beltran-Parrazal L; Department of Neurology, UCLA School of Medicine, 710 Westwood Plaza, Los Angeles, CA 90095-1769, USA.; Charles A

Subjects: Action Potentials/Action Potentials/Action Potentials/*drug effects ; Calcium Signaling/Calcium Signaling/Calcium Signaling/*drug effects ; Potassium Channels/Potassium Channels/Potassium Channels/*metabolism

  • Source: British journal of pharmacology [Br J Pharmacol] 2003 Nov; Vol. 140 (5), pp. 881-8. Date of Electronic Publication: 2003 Oct 06.Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print-Electronic Cited Medium: Print ISSN: 0007-1188 (Print)

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