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Academic Journal

Development of Kinase Inhibitors via Metal-Catalyzed C–H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies

Subjects: DYRK1A; CDK5; protein kinases

  • Source: ISSN: 1420-3049 ; Molecules ; https://normandie-univ.hal.science/hal-02024491 ; Molecules, 2018, 23 (9), pp.2181. ⟨10.3390/molecules23092181⟩.

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Academic Journal

Development of Kinase Inhibitors via Metal-Catalyzed C–H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies

Subjects: DYRK1A; CDK5; protein kinases

  • Source: ISSN: 1420-3049 ; Molecules ; https://normandie-univ.hal.science/hal-02024491 ; Molecules, 2018, 23 (9), pp.2181. ⟨10.3390/molecules23092181⟩.

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Academic Journal

Development of Kinase Inhibitors via Metal-Catalyzed C–H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies

Subjects: DYRK1A; CDK5; protein kinases

  • Source: ISSN: 1420-3049 ; Molecules ; https://normandie-univ.hal.science/hal-02024491 ; Molecules, 2018, 23 (9), pp.2181. ⟨10.3390/molecules23092181⟩.

تفاصيل العنوان

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Academic Journal

Development of Kinase Inhibitors via Metal-Catalyzed C–H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies

Subjects: DYRK1A; CDK5; protein kinases

  • Source: ISSN: 1420-3049 ; Molecules ; https://normandie-univ.hal.science/hal-02024491 ; Molecules, 2018, 23 (9), pp.2181. ⟨10.3390/molecules23092181⟩.

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Academic Journal

Development of Kinase Inhibitors via Metal-Catalyzed C–H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies

Subjects: CLK1; protein kinases; CDK5

  • Source: ISSN: 1420-3049 ; Molecules ; https://hal-normandie-univ.archives-ouvertes.fr/hal-02024491 ; Molecules, MDPI, 2018, 23 (9), pp.2181. ⟨10.3390/molecules23092181⟩.

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Academic Journal

Development of Kinase Inhibitors via Metal-Catalyzed C–H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies

Subjects: DYRK1A; CDK5; protein kinases

  • Source: ISSN: 1420-3049 ; Molecules ; https://normandie-univ.hal.science/hal-02024491 ; Molecules, 2018, 23 (9), pp.2181. ⟨10.3390/molecules23092181⟩.

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Academic Journal

Synthesis of bioactive 2-(arylamino)thiazolo[5,4-f]-quinazolin-9-ones via the Hügershoff reaction or Cu- catalyzed intramolecular C-S bond formation

Subjects: CLK1; CK1; Hügershoff reaction

  • Source: ISSN: 1420-3049 ; Molecules ; https://normandie-univ.hal.science/hal-02046212 ; Molecules, 2016, 21 (6), pp.794. ⟨10.3390/molecules21060794⟩.

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Academic Journal

Synthesis of Thiazolo[5,4-f]quinazolin-9(8H)-ones as Multi-Target Directed Ligands of Ser/Thr Kinases

Subjects: 4-f ]quinazolin-9(8H)-ones; thiazolo[5; CLK1

  • Source: ISSN: 1420-3049 ; Molecules ; https://normandie-univ.hal.science/hal-02046213 ; Molecules, 2016, 21 (5), pp.578. ⟨10.3390/molecules21050578⟩.

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